Acetaminophen, alfentanil, alfuzosin, almotriptan, alprazolam, amiodarone, amlodipine, aprepitant, astemizole, atazanavir, atorvastatin, bepridil, bexarotene, bosentan, bromocriptine, budesonide, buspirone, carbamazepine, cisapride, clarithromycin, clonazepam, clopidogrel, cocaine, colchicine, conivaptan, cortisol, cyclosporine, dapsone, darunavir, dasatinib, delavirdine, dexamethasone, diazepam, dihydroergotamine, dihydropyridines, diltiazem, disopyramide, doxorubicin, droperidol, dutasteride, ebastine, efavirenz, eletriptan, eplerenone, ergotamine, erlotinib, erythromycin, estazolam, eszopiclone, ethinyl estradiol, ethosuximide, etoposide, everolimus, exemestane, felodipine, fentanyl, finasteride, flurazepam, fluticasone, fosamprenavir, galantamine, gefitinib, gestodene, granisetron, halofantrine, ifosfamide, imatinib, indinavir, irinotecan, isradipine, itraconazole, ixabepilone, lapatinib, lidocaine, loperamide, lopinavir, loratadine, lovastatin, macrolides, maraviroc, mefloquine, methadone, methylprednisolone, miconazole, midazolam, mifepristone, modafinil, nefazodone, nevirapine, nicardipine, nifedipine, nimodipine, nisoldipine, paclitaxel, paricalcitol, pimozide, pioglitazone, praziquantel, prednisolone, prednisone, progesterone, quetiapine, quinacrine, quinidine, quinine, ranolazine, rapamycin, repaglinide, rifabutin, ritonavir, saquinavir, sibutramine, sildenafil, simvastatin, sirolimus, solifenacin, spironolactone, sufentanil, sulfamethoxazole, sunitinib, tacrolimus, tadalafil, tamoxifen, tamsulosin, teniposide, terfenadine, testosterone, tetrahydrocannabinol, tiagabine, tinidazole, tipranavir, tolvaptan, topiramate, triazolam, troleandomycin, vardenafil, verapamil, vinblastine, vincristine, ziprasidone, zolpidem, zonisamide, zopiclone Amprenavir, azamulin, boceprevir, clarithromycin, conivaptan, diltiazem, erythromycin, fluconazole, grapefruit juice (furanocoumarins), indinavir, itraconazole, ketoconazole, lopinavir, mibefradil, nefazodone, nelfinavir, posaconazole, ritonavir, saquinavir, telaprevir, telithromycin, troleandomycin, verapamil, voriconazole 1CYP3A5 has similar substrate and inhibitor profiles but, except for a few drugs, is generally less active than CYP3A4.